本發明係有關於一抑制冠狀病毒之醫藥組合物,其中包括一種或多種選自本發明所述群組之化合物(包括其醫藥上可接受之鹽類以及前驅藥物);本發明亦提供一醫藥用套組,包括有一容器,一種或多種保存於容器中之如上述化合物,以及一附帶於容器之標示(如一標籤或是一夾頁),用以說明化合物對於抑制冠狀病毒之使用方法。A pharmaceutical composition and packaged product for inhibiting coronavirus infection is disclosed. The composition includes at least one compounds (as well as their pharmaceutically acceptable salts and prodrugs) as described in present invention. The packaged product, comprising a container; a compound selected from present invention and; a legend associated with the container and indicating administration of the compound for treating coronavirus infection.