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Showing items 51-75 of 142. (6 Page(s) Totally) << < 1 2 3 4 5 6 > >> View [10|25|50] records per page

Date	Title	Relation
2014-07	Anaplastic lymphoma kinase (ALK) inhibitors: A review of design and discovery	MedChemComm. 2014 Jul;5(9):1266-1279.
2014-05	Facile identification of dual FLT3-Aurora A inhibitors: A computer-guided drug design approach	ChemMedChem. 2014 May;9(5):953-961.
2014-05	Cover Picture: Facile identification of dual FLT3–aurora a inhibitors: A computer-guided drug design approach (ChemMedChem 5/2014)	ChemMedChem. 2014 May;9(5):861.
2013-09-22	A novel Aurora-A inhibitor, BPR1K0609S1, sensitizes colorectal tumor cells to 5-fluorofracil (5-FU) treatment [Erratum:International Journal of Biological Sciences. 2013 Apr 29;9(4):403-411]	International Journal of Biological Sciences. 2013 Sep 22;9(9):947.
2013-07-25	Pronounced induction of endoplasmic reticulum stress and tumor suppression by surfactant-free poly(lactic-co-glycolic acid) nanoparticles via modulation of the PI3K signaling pathway	International Journal of Nanomedicine. 2013 Jul 25;2013(8):2689-2707.
2013-06-28	Optimization of ligand and lipophilic efficiency to identify an in vivo active furano-pyrimidine aurora kinase inhibitor	Journal of Medicinal Chemistry. 2013 Jun 28;56(13):5247-5260.
2013-06	An antimitotic and antivascular agent BPR0L075 overcomes multidrug resistance and induces mitotic catastrophe in paclitaxel-resistant ovarian cancer cells	PLoS ONE. 2013 Jun;8(6):Article number e65686.
2013-05	Aurora kinase inhibitors reveal mechanisms of HURP in nucleation of centrosomal and kinetochore microtubules	Proceedings of the National Academy of Sciences of the United States of America. 2013 May;110(19):E1779-E1787.
2013-05	Protein kinase inhibitor design by targeting the Asp-Phe-Gly (DFG) motif: The role of the DFG motif in the design of epidermal growth factor receptor inhibitors	Journal of Medicinal Chemistry. 2013 May;56(10):3889-3903.
2013-04-29	A novel Aurora-A inhibitor, BPR1K0609S1, sensitizes colorectal tumor cells to 5-fluorofracil (5-FU) treatment	International Journal of Biological Sciences. 2013 Apr 29;9(4):403-411.
2013-02-20	Parallel screening of Wild-Type and drug-resistant targets for anti-resistance neuraminidase inhibitors	PLoS ONE. 2013 Feb 20;8(2):Article number e56704.
2013-01	3D-QSAR-assisted drug design: Identification of a potent quinazoline-based aurora kinase inhibitor	ChemMedChem. 2013 Jan;8(1):136-148.
2013-01	Substituent effects on the photorearrangements of unsymmetrically substituted diazinobarrelenes	RSC Advances. 2013 Jan;3(4):1165-1178.
2012-12	An efficient, mild and scalable synthesis of bioactive compounds containing the angelicin scaffold	Journal of the Chinese Chemical Society. 2012 Dec;59(12):1548-1554.
2012-09	Anti-influenza drug discovery: Identification of an orally bioavailable quinoline derivative through activity- and property-guided lead optimization	ChemMedChem. 2012 Sep;7(9):1546-1550.
2012-08-24	Tubulin-destabilizing agent BPR0L075 induces vascular-disruption in human breast cancer mammary fat pad xenografts	PLoS ONE. 2012 Aug 24;7(8):Article number e43314.
2012-02	Identification of BPR3P0128 as an Inhibitor of cap-snatching activities of influenza virus	Antimicrobial Agents and Chemotherapy. 2012 Feb;56(2):647-657.
2012-01	A High-throughput cell-based screening for L858R/T790M mutant epidermal growth factor receptor inhibitors	Anticancer Research. 2012 Jan;32(1):147-151.
2011-09	Synthesis and biological evaluation of 1-(4′-Indolyl and 6′-Quinolinyl) indoles as a new class of potent anticancer agents	European Journal of Medicinal Chemistry. 2011 Sep;46(9):3623-3629.
2011-09	Inhibition of HIV-1 Tat-mediated transcription by a coumarin derivative, BPRHIV001, through the Akt pathway	Journal of Virology. 2011 Sep;85(17):9114-9126
2011-08	BPR1K653, a novel aurora kinase inhibitor, exhibits potent anti-proliferative activity in MDR1 (P-gp170)-mediated multidrug-resistant cancer cells	PLoS ONE. 2011 Aug;6(8):Article number e23485.
2011-06	Aurora kinase inhibitor patents and agents in clinical testing: an update (2009-10)	Expert Opinion on Therapeutic Patents. 2011 Jun;21(6):857-884.
2011-04-28	Scaffold-hopping strategy: Synthesis and biological evaluation of 5,6-Fused bicyclic heteroaromatics to identify orally bioavailable anticancer agents	Journal of Medicinal Chemistry. 2011 Apr 28;54(8):3076-3080.
2011-03-07	2-Amino-3,4,5-Trimethoxybenzophenones as Potent Tubulin Polymerization Inhibitors	ChemMedChem. 2011 Mar 7;6(3):450-456.
2010-10-28	Design and synthesis of tetrahydropyridothieno[2,3-d]pyrimidine scaffold based epidermal growth factor receptor (EGFR) kinase inhibitors: the role of side chain chirality and michael acceptor group for maximal potency	Journal of Medicinal Chemistry. 2010 Oct 28;53(20):7316-7326.

Showing items 51-75 of 142. (6 Page(s) Totally) << < 1 2 3 4 5 6 > >> View [10|25|50] records per page