2024-04 |
Design, synthesis, and anticancer evaluation of 1-benzo[1,3]dioxol-5-yl-3-N-fused heteroaryl indoles |
Molecular Diversity. 2024 Apr;28(2):595-608. |
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2024-01-23 |
Decrypting orphan GPCR drug discovery via multitask learning |
Journal of Cheminformatics. 2024 Jan 23;16:Article number 10. |
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2023-10-05 |
Discovery of tetrasubstituted thiophenes as Cisd2 activators: A potential novel therapeutic option in nonalcoholic fatty liver disease |
European Journal of Medicinal Chemistry. 2023 Oct 05;258:Article number 115583. |
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2023-03-17 |
A convenient diels-alder approach toward potential polyketide-like antibiotics using alpha-activated alpha,Beta-unsaturated 4,4-dimethyl-1-tetralones as dienophiles |
Molecules. 2023 Mar 17;28(6):Article number 2739. |
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2022-03-02 |
Discovery of potential neuroprotective agents against paclitaxel-induced peripheral neuropathy |
Journal of Medicinal Chemistry. 2022 Mar 2;65(6):4767-4782. |
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2020-02 |
Design, synthesis and anticancer evaluation of beta-carboline-1-one hydantoins |
Future Medicinal Chemistry. 2020 Feb;12(3):183-192. |
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2020-01-01 |
Delayed intervention with a novel SGLT2 inhibitor NGI001 suppresses diet-induced metabolic dysfunction and nonalcoholic fatty liver disease in mice |
British Journal of Pharmacology. 2020 Jan 1;177(2):239-253. |
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2019-03 |
Synthesis and biological evaluation of N-glucosyl indole derivatives as sodium-dependent glucose co-transporter 2 inhibitors |
Bioorganic Chemistry. 2019 Mar;83:520-525. |
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2018-01-01 |
Identification of an oxime-containing C-glucosylarene as a potential inhibitor of sodium-dependent glucose co-transporter 2 |
European Journal of Medicinal Chemistry. 2018 Jan 1;143:611-620. |
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2016-12-08 |
Bromomethylthioindole inspired carbazole hybrids as promising class of anti-MRSA agents |
ACS Medicinal Chemistry Letters. 2016 Dec 8;7(12):1191-1196. |
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2016-09 |
Mycotoxin patulin suppresses innate immune responses by mitochondrial dysfunction and p62/sequestosome-1-dependent mitophagy |
Journal of Biological Chemistry. 2016 Sep;291(37):19299-19311. |
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2016-07 |
Total synthesis of the naturally occurring glycosylflavone aciculatin |
Journal of Natural Products. 2016 Jul;79(7):1719-1723. |
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2016-05 |
N-Indolylglycosides bearing modifications at the glucose C6-Position as Sodium-Dependent Glucose Co-transporter 2 inhibitors |
Bioorganic and Medicinal Chemistry. 2016 May;24(10):2242-2250. |
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2015-08 |
Optimization of furanopyrimidine-based kinase inhibitors: Identification of a BTK kinase inhibitor for the treatment of B cell lymphoma |
Abstracts of Papers of the American Chemical Society. 2015 Aug;250:Meeting Abstract 180. |
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2015-07 |
Development and application of a fluorescent glucose uptake assay for the high-throughput screening of non-glycoside SGLT2 inhibitors |
European Journal of Pharmaceutical Sciences. 2015 Jul;74:40-44. |
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2014-09 |
N-Iodosuccinimide and acid-washed molecular sieves (NIS/AW-300 MS) as promoters in thioglycoside activation |
Tetrahedron. 2014 Sep;70(38):6757-6762. |
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2014-08 |
Discovery of selective inhibitors of Glutaminase-2, which inhibit mTORC1, activate autophagy and inhibit proliferation in cancer cells |
Oncotarget. 2014 Aug;5(15):6087-6101. |
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2014-04-15 |
Glycoside compounds |
US8697658B2/2014-04-15 |
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2012-09 |
Synthesis and biological evaluation of novel C-indolylxylosides as sodium-dependent glucose co-transporter 2 inhibitors |
European Journal of Medicinal Chemistry. 2012 Sep;55:32-38. |
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2011-08 |
Colloid-based multiplexed screening for plant biomass-degrading glycoside hydrolase activities in microbial communities |
Energy and Environmental Science. 2011 Aug;4(8):2884-2893. |
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2011-07-25 |
The first total synthesis of cytopiloyne, an anti-diabetic, polyacetylenic glucoside |
Chemistry-A European Journal. 2011 Jul 25;17(31):8696-8703. |
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2011-06 |
Development of sodium-dependent glucose co-transporter 2 inhibitors as potential anti-diabetic therapeutics |
Current Topics In Medicinal Chemistry. 2011 Jun;11(12):1476-1512. |
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2011-01-13 |
Discovery of novel N -Beta- d -Xylosylindole derivatives as sodium-dependent glucose cotransporter 2 (SGLT2) inhibitors for the management of hyperglycemia in diabetes |
Journal of Medicinal Chemistry. 2011 Jan 13;54(1):166-178. |
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2010-12 |
Discovery of non-glycoside sodium-dependent glucose Co-transporter 2 (SGLT2) inhibitors by ligand-based virtual screening |
Journal of Medicinal Chemistry. 2010 Dec;53(24):8770-8774. |
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