| 2016-12 |
Phenyl benzenesulfonylhydrazides: Selective indoleamine 2,3-dioxygenase inhibitors with potent in vivo pharmacodynamic activity and antitumor efficacy |
European Journal of Cancer. 2016 Dec;68(Suppl. 1):S83-S84. |
 |
| 2016-12 |
Novel cKIT kinase inhibitor, BPRCKJ001, as an advanced therapeutic candidate for GIST |
Annals of Oncology. 2016 Dec;27(Suppl. 9):Meeting Abstract 2P. |
|
| 2016-11-29 |
Discovery of novel inhibitors of Aurora kinases with indazole scaffold: In silico fragment-based and knowledge-based drug design |
European Journal of Medicinal Chemistry. 2016 Nov 29;124:186-199. |
|
| 2016-11-18 |
Cobalt(II)-catalyzed aerobic oxidation of terminal-capped alkynyl alpha-cyano alkanone systems. An oxygen-mediated radical chain reaction |
Journal of Organic Chemistry. 2016 Nov 18;81(22):10759-10768. |
|
| 2016-10 |
Cytotoxic cardenolides and sesquiterpenoids from the fruits of Reevesia formosana |
Phytochemistry. 2016 Oct;130:282-290. |
|
| 2016-10 |
BPR1J373, an oral multiple tyrosine kinase inhibitor, targets c-KIT for the treatment of c-KIT driven myeloid leukemia |
Molecular Cancer Therapeutics. 2016 Oct;15(10):2323-2333. |
|
| 2016-10 |
Multifunctional nanoparticles for oral protein drug delivery |
Diabetes Research and Clinical Practice. 2016 Oct;120(Suppl. 1):S19. |
|
| 2016-09 |
Mycotoxin patulin suppresses innate immune responses by mitochondrial dysfunction and p62/sequestosome-1-dependent mitophagy |
Journal of Biological Chemistry. 2016 Sep;291(37):19299-19311. |
|
| 2016-09 |
Activation of delta-opioid receptor contributes to the antinociceptive effect of oxycodone in mice |
Pharmacological Research. 2016 Sep;111:867-876. |
|
| 2016-08 |
Desferal regulates hCtr1 and transferrin receptor expression through Sp1 and exhibits synergistic cytotoxicity with platinum drugs in oxaliplatin-resistant human cervical cancer cells in vitro and in vivo |
Oncotarget. 2016 Aug;7(31):49310-49321. |
|
| 2016-08 |
Dipeptidyl peptidase-4 inhibitor LAF-237 improves glucose tolerance and expends graft beta cell mass in diabetic mice transplanted with a sufficient number of islets |
Diabetologia. 2016 Aug;59(Suppl. 1):S198. |
|
| 2016-07-28 |
Design and synthesis of 1,2,3-triazole-containing N-acyl zanamivir analogs as potent neuraminidase inhibitors |
European Journal of Medicinal Chemistry. 2016 Jul 28;123:397-406. |
|
| 2016-07-22 |
Orexins contribute to restraint stress-induced cocaine relapse by endocannabinoid-mediated disinhibition of dopaminergic neurons |
Nature Communications. 2016 Jul 22;7:Article number 12199. |
|
| 2016-07-01 |
MPT0B098, a microtubule inhibitor, suppresses JAK2/STAT3 signaling pathway through modulation of SOCS3 stability in oral squamous cell carcinoma |
PLoS ONE. 2016 Jul 1;11(7):Article number e0158440. |
|
| 2016-07 |
In vitro and in vivo studies of a potent capsid-binding inhibitor of enterovirus 71 |
Journal of Antimicrobial Chemotherapy. 2016 Jul;71(7):1922-1932. |
|
| 2016-07 |
Therapeutic polymeric nanoparticles and the methods of making and using thereof: A patent evaluation of WO2015036792 |
Expert Opinion on Therapeutic Patents. 2016 Jul;26(7):751-755. |
|
| 2016-07 |
Total synthesis of the naturally occurring glycosylflavone aciculatin |
Journal of Natural Products. 2016 Jul;79(7):1719-1723. |
|
| 2016-06 |
The sigma-1 receptor-zinc finger protein 179 pathway protects against hydrogen peroxide-induced cell injury |
Neuropharmacology. 2016 Jun;105:1-9. |
|
| 2016-05-19 |
Non-small-cell lung cancer cells combat epidermal growth factor receptor tyrosine kinase inhibition through immediate adhesion-related responses |
OncoTargets and Therapy. 2016 May 19;9:2961-2973. |
|
| 2016-05 |
N-Indolylglycosides bearing modifications at the glucose C6-Position as Sodium-Dependent Glucose Co-transporter 2 inhibitors |
Bioorganic and Medicinal Chemistry. 2016 May;24(10):2242-2250. |
|
| 2016-05 |
An early granulocyte colony-stimulating factor treatment attenuates neuropathic pain through activation of mu opioid receptors on the injured nerve |
Scientific Reports. 2016 May;6:Article number 25490. |
|
| 2016-04-12 |
Pyrazolylamine derivatives reveal the conformational switching between type I and type II binding modes of Anaplastic Lymphoma Kinase (ALK) |
Journal of Medicinal Chemistry. 2016 Apr 12;59(8):3906-3919. |
|
| 2016-04 |
Discovery and development of tylophorine derived dibenzoquinolines-33b compounds into therapeutic agents |
The FASEB Journal. 2016 Apr;30(1, Suppl.):Meeting Abstract lb56. |
 |
| 2016-03 |
Probing for improved selectivity with dipeptide-derived inhibitors of dipeptidyl peptidases 8 and 9: The impact of P1-variation |
MedChemComm. 2016 Mar;7(3):433-438. |
|
| 2016-03 |
Disruption of protein-protein interactions: Hot spot detection, structure-based virtual screening and in vitro testing for the anti-cancer drug target survivin |
RSC Advances. 2016 Mar;6(38):31947-31959. |
|
